{"product_id":"tirzepatide","title":"Tirzepatide","description":"\u003ch2\u003eTirzepatide\u003c\/h2\u003e\n\u003cp\u003eTirzepatide is a synthetic 39-amino acid dual agonist peptide targeting both the glucose-dependent insulinotropic polypeptide (GIP) receptor and the glucagon-like peptide-1 (GLP-1) receptor. Originally developed as a novel approach to metabolic disease research, tirzepatide has attracted significant scientific interest for its dual incretin mechanism, which distinguishes it from single-receptor GLP-1 agonists. It is supplied here as a lyophilised research compound for in vitro and preclinical investigation.\u003c\/p\u003e\n\u003ch3\u003eMechanism of Action\u003c\/h3\u003e\n\u003cp\u003eTirzepatide acts as a co-agonist at GIP (GIPR) and GLP-1 (GLP-1R) receptors, both of which are G-protein-coupled receptors that signal via cAMP elevation. GLP-1R activation enhances glucose-dependent insulin secretion and suppresses glucagon release, while GIPR activation contributes additional insulinotropic and potentially adipose-regulatory effects. The dual agonism is hypothesised to produce synergistic metabolic effects beyond those achievable with GLP-1 monotherapy, making tirzepatide a key subject in obesity, insulin resistance, and metabolic syndrome research.\u003c\/p\u003e\n\u003ch3\u003eResearch Applications\u003c\/h3\u003e\n\u003cul\u003e\n\u003cli\u003eDual GIP\/GLP-1 receptor pharmacology studies\u003c\/li\u003e\n\u003cli\u003eInsulin secretion and glucose homeostasis modelling\u003c\/li\u003e\n\u003cli\u003eObesity and adipose tissue metabolism research\u003c\/li\u003e\n\u003cli\u003eIncretin biology and pancreatic beta-cell function investigation\u003c\/li\u003e\n\u003cli\u003eMetabolic syndrome and insulin resistance preclinical models\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003ch3\u003eSpecifications\u003c\/h3\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cstrong\u003eMolecular Formula:\u003c\/strong\u003e \u003cmeta charset=\"utf-8\"\u003eC₂₂₅H₃₄₈N₄₈O₆₈\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eMolecular Weight:\u003c\/strong\u003e 4813.5 g\/mol\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eCAS Number:\u003c\/strong\u003e 2023788-19-2\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003ePurity:\u003c\/strong\u003e ≥98%\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eForm:\u003c\/strong\u003e Lyophilised powder\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eStorage:\u003c\/strong\u003e -20°C\u003c\/li\u003e\n\u003cli\u003e\n\u003cstrong\u003eShelf Life:\u003c\/strong\u003e 24 months\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp\u003e\u003cem\u003eThis product is intended for legitimate laboratory and analytical research use only. Not for diagnostic, therapeutic, or consumer use.\u003c\/em\u003e\u003c\/p\u003e","brand":"Vanta Labs","offers":[{"title":"5mg","offer_id":58103432380680,"sku":"TIRZE-5MG","price":21.99,"currency_code":"GBP","in_stock":true},{"title":"10mg","offer_id":58103432413448,"sku":"TIRZE-10MG","price":44.99,"currency_code":"GBP","in_stock":true},{"title":"15mg","offer_id":58103432446216,"sku":"TIRZE-15MG","price":55.99,"currency_code":"GBP","in_stock":true},{"title":"20mg","offer_id":58103432478984,"sku":"TIRZE-20MG","price":63.99,"currency_code":"GBP","in_stock":true},{"title":"30mg","offer_id":58103432511752,"sku":"TIRZE-30MG","price":80.99,"currency_code":"GBP","in_stock":true},{"title":"40mg","offer_id":58103432544520,"sku":"TIRZE-40MG","price":99.99,"currency_code":"GBP","in_stock":true},{"title":"60mg","offer_id":58103432577288,"sku":"TIRZE-60MG","price":139.99,"currency_code":"GBP","in_stock":true},{"title":"90mg","offer_id":58103432610056,"sku":"TIRZE-90MG","price":159.99,"currency_code":"GBP","in_stock":true},{"title":"100mg","offer_id":58103432642824,"sku":"TIRZE-100MG","price":199.99,"currency_code":"GBP","in_stock":true},{"title":"120mg","offer_id":58103432675592,"sku":"TIRZE-120MG","price":230.99,"currency_code":"GBP","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/1049\/8886\/8872\/files\/tirzepatide.png?v=1782892821","url":"https:\/\/vantalabsuk.com\/products\/tirzepatide","provider":"Vanta Labs","version":"1.0","type":"link"}